ORIGINAL RESEARCH ARTICLES

Cardiovascular Safety of VIAN-c4551, an Antiangiogenic Peptide Derived From Vasoinhibin
Miguel A. García-González, Alejandro D. Miguel-Martínez, Abimael González-Hernández, Magdalena Zamora, Elva Adán-Castro, Xarubet Ruíz-Herrera, María A. Carbajo-Mata, Jakob Triebel, Thomas Bertsch, José G. Lopez-Lopez, Gonzalo Martínez de la Escalera, Juan Pablo Robles, Carmen Clapp, Carlos M. Villalón
Drug Development Research 2025 · Journal article ↗ · PDF ↗
Relationships Between H2S and OT/OTR Systems in Preeclampsia
Tamara Merz, Sarah Ecker, Nicole Denoix, Oscar McCook, Stefanie Kranz, Ulrich Wachter, Edit Rottler, Thomas Papadopoulos, Christoph Fusch, Cosima Brucker, Jakob Triebel, Thomas Bertsch, Peter Radermacher, Christiane Waller
Antioxidants 2025 (Basel) · Journal article ↗ · PDF ↗
Topical eye administration of the antiangiogenic peptide VIAN-c4551 protects against experimental diabetic macular edema
Adan-Castro E, Zamora M, Granados-Carrasco D, Siqueiros-Márquez L, García-Rodrigo JF, Bertsch T, Triebel J, Martínez de la Escalera G, Robles JP, Clapp C.
Scientific Reports 2025 · Journal article ↗ · PDF ↗
The antiangiogenic peptide VIAN-c4551 inhibits lung melanoma metastasis in mice by reducing pulmonary vascular permeability
Perez AL, Zamora M, Bahena M, Aramburo-Williams R, Adan-Castro E, Granados-Carrasco D, Bertsch T, Triebel J, Martinez de la Escalera G, Robles JP, Clapp C.
PLoS One 2025 · Journal article ↗ · PDF ↗
Vasoinhibin is Generated by the Renin-angiotensin System
Francisco Freinet Núñez, Lourdes Siqueiros-Marquez, Elva Adán-Castro, Magdalena Zamora, Juan Pablo Robles, Xarubet Ruíz-Herrera, Thomas Bertsch, Jakob Triebel, Gonzalo Martínez de la Escalera, Carmen Clapp
Endocrinology 2025 · Journal article ↗ · PDF ↗
Mass Spectrometric and Immunologic Detection of Prolactin-Derived Vasoinhibin in Human Serum
Jakob Triebel, David Harris, Nils Davies, Johannes Ebnet, Leon Neugebauer, Christin Friedrich, Hülya Markl-Hahn, Hans-Herbert Steiner, Thomas Bertsch
Clinical Laboratory 2024 · Journal article ↗ · PDF ↗
Immunometric and Functional Measurement of Endogenous Vasoinhibin in Human Sera
Magdalena Zamora, David Harris, Nils Davies, Johannes Ebnet, Peter Radermacher, Cosima Brucker, Christiane Waller, Juan Pablo Robles, Thomas Bertsch, Carmen Clapp, Jakob Triebel
Frontiers in Endocrinology (Lausanne) 2024 · Journal article ↗ · PDF ↗
Levosulpiride for the treatment of diabetic macular oedema: a phase 2 randomized clinical trial
Carlos D Núñez-Amaro, Mariana López, Elva Adán-Castro, Ma Ludivina Robles-Osorio, Renata García-Franco, Marlon García-Roa, Yolanda Villalpando-Gómez, Paulina Ramírez-Neria, Nayeli Pineiro, Juan Fernando Rubio-Mijangos, Jorge Sánchez, Gabriela Ramírez-Hernández, Lourdes Siqueiros-Márquez, Nundehui Díaz-Lezama, Ellery López-Star, Thomas Bertsch, Gonzalo Marínez de la Escalera, Jakob Triebel, Carmen Clapp
Eye (London) 2023 · Journal article ↗ · PDF ↗
Vasoinhibin’s Apoptotic, Inflammatory, and Fibrinolytic Actions Are in a Motif Different From Its Antiangiogenic HGR Motif
Juan Pablo Robles, Magdalena Zamora, Jose F. Garcia-Rodrigo, Alma Lorena Perez, Thomas Bertsch, Gonzalo Martinez de la Escalera, Jakob Triebel, Carmen Clapp
Endocrinology 2023 · Journal article ↗ · PDF ↗
Human Placental Tissue Contains a Placental Lactogen Derived Vasoinhibin
Hülya Markl-Hahn, Leon Neugebauer, Livia Lenke, Sarah Ecker, Tamara Merz, Oscar McCook, Noura Khoder, Cosima Brucker, Peter Radermacher, Christiane Waller, Carmen Clapp, Thomas Bertsch, Jakob Triebel
Journal of the Endocrine Society 2022 · Journal article ↗ · PDF ↗
A Comparative Phylogenetic Analysis of Prolactin Cleavage Sites for the Generation of Vasoinhibin In Vertebrates
Andreas Leuchs, Nils Davies, Christin Friedrich, Sabrina Trier, Carmen Clapp, Thomas Bertsch, Jakob Triebel
General and Comparative Endocrinology 2022 · Journal article ↗ · PDF ↗
Sulpiride-induced hyperprolactinaemia increases retinal vasoinhibin and protects against diabetic retinopathy in rats
Elva Adán-Castro, Lourdes Siqueiros-Márquez, Gabriela Ramírez-Hernández, Nundehui Díaz-Lezama, Xarubet Ruíz-Herrera, Francisco Freinet Núñez, Carlos D. Núñez-Amaro, Ma. Ludivina Robles-Osorio, Thomas Bertsch, Jakob Triebel, Gonzalo Martínez de la Escalera, Carmen Clapp
Journal of Neuroendocrinology 2022 · Journal article ↗
Complement Proteins C5/C5a, Cathepsin D and Prolactin in Chondrocytes: A Possible Crosstalk in the Pathogenesis of Osteoarthritis
Sandeep Silawal, Miriam Wagner, Dominik Roth, Thomas Bertsch, Silke Schwarz, Maximilian Willauschus, Markus Gesslein, Jakob Triebel, Gundula Schulze-Tanzil
Cells 2022 · Journal article ↗ · PDF ↗
Plasmin generates vasoinhibin-like peptides by cleaving prolactin and placental lactogen
Christin Friedrich, Leon Neugebauer, Magdalena Zamora, Juan Pablo Robles, Gonzalo Martínez de la Escalera, Carmen Clapp, Thomas Bertsch, Jakob Triebel
Molecular and Cellular Endocrinology 2021 · Journal article ↗ · PDF ↗
Development of Vasoinhibin-specific Monoclonal Antibodies
Nils Müller, Juan Pablo Robles, Magdalena Zamora, Johannes Ebnet, Hülya Markl-Hahn, Gonzalo Martínez de la Escalera, Carmen Clapp, Thomas Bertsch, Jakob Triebel
Frontiers in Endocrinology (Lausanne) 2021 · Journal article ↗ · PDF ↗
Thrombin Cleaves Prolactin Into a Potent 5.6-kDa Vasoinhibin: Implication for Tissue Repair
Magdalena Zamora, Juan Pablo Robles, Manuel B Aguilar, Sergio de Jesús Romero-Gómez, Thomas Bertsch, Gonzalo Martínez de la Escalera, Jakob Triebel, Carmen Clapp
Endocrinology 2021 · Journal article ↗
The HGR motif is the antiangiogenic determinant of vasoinhibin: implications for a therapeutic orally active oligopeptide
Juan Pablo Robles · Magdalena Zamora · Lourdes Siqueiros‑Marquez · Elva Adan‑Castro · Gabriela Ramirez‑Hernandez · Francisco Freinet Nuñez · Fernando Lopez‑Casillas · Robert P. Millar Thomas Bertsch · Gonzalo Martínez de la Escalera · Jakob Triebel · Carmen Clapp
Angiogenesis 2021 · Journal article ↗ · PDF ↗
Levosulpiride Increases the Levels of Prolactin and Antiangiogenic Vasoinhibin in the Vitreous of Patients with Proliferative Diabetic Retinopathy
Carlos D. Nuñez-Amaro; Aura Ileana Moreno-Vega; Elva Adan-Castro; Magdalena Zamora; Renata Garcia-Franco; Paulina Ramirez-Neria; Marlon Garcia-Roa; Yolanda Villalpando; Juan Pablo Robles; Gabriela Ramirez-Hernandez; Mariana Lopez; Jorge Sanchez; Ellery Lopez-Star; Thomas Bertsch; Gonzalo Martinez de la Escalera; Ma. Ludivina Robles-Osorio; Jakob Triebel; Carmen Clapp
Translational Vision Science and Technology 2020 · Journal article ↗ · PDF ↗
Matrix Metalloproteases and Cathepsin D in Human Serum do not Cleave Prolactin to Generate Vasoinhibin
Jakob Triebel, Nicole Schauer, Magdalena Zamora, Aura Ileana Moreno-Vega, Gonzalo Martínez de la Escalera, Carmen Clapp, Thomas Bertsch
Clinical Laboratory 2020 · Journal article ↗ · PDF ↗
Improving Immunotherapy Against B-Cell Malignancies Using gammadelta T-Cell-specific Stimulation and Therapeutic Monoclonal Antibodies
Hoeres, T., Pretscher, D., Holzmann, E., Smetak, M., Birkmann, J., Triebel, J., Bertsch, T., Wilhelm, M.
Journal of Immunotherapy 2019 · Journal article ↗
Vasoinhibin comprises a three-helix bundle and its antiangiogenic domain is located within the first 79 residues
Juan Pablo Robles, Magdalena Zamora, José Luis Velasco-Bolom, Miriam Tovar, Ramón Garduño-Juárez, Thomas Bertsch, Gonzalo Martínez de la Escalera, Jakob Triebel & Carmen Clapp
Scientific Reports 2018 · Journal article ↗ · PDF ↗
Basis and Design of a Randomized Clinical Trial to Evaluate the Effect of Levosulpiride on Retinal Alterations in Patients With Diabetic Retinopathy and Diabetic Macular Edema
Robles-Osorio, M. L., R. Garcia-Franco, C. D. Nunez-Amaro, X. Mira-Lorenzo, P. Ramirez-Neria, W. Hernandez, E. Lopez-Star, T. Bertsch, G. Martinez de la Escalera, J. Triebel and C. Clapp
Frontiers in Endocrinology (Lausanne) 2018 · Journal article ↗ · PDF ↗
Human Prolactin Point Mutations and Their Projected Effect on Vasoinhibin Generation and Vasoinhibin-Related Diseases
Jakob Triebel, Christin Friedrich, Andreas Leuchs, Gonzalo Martínez de la Escalera, Carmen Clapp, Thomas Bertsch
Frontiers in Endocrinology (Lausanne) 2017 · Journal article ↗ · PDF ↗
Higher prolactin and vasoinhibin serum levels associated with incidence and progression of retinopathy of prematurity
Zepeda-Romero, L. C., M. Vazquez-Membrillo, E. Adan-Castro, F. Gomez-Aguayo, J. A. Gutierrez-Padilla, E. Angulo-Castellanos, J. C. Barrera de Leon, C. Gonzalez-Bernal, M. A. Quezada-Chalita, A. Meza-Anguiano, N. Diaz-Lezama, G. Martinez de la Escalera, J. Triebel and C. Clapp
Pediatric Research 2017 · Journal article ↗ · PDF ↗
Percutaneous Closure of Left Atrial Appendage affects Mid-Term Release of MR-proANP
Behnes, M., B. Sartorius, A. Wenke, S. Lang, U. Hoffmann, C. Fastner, M. Borggrefe, T. Roth, J. Triebel, T. Bertsch and I. Akin
Scientific Reports 2017 · Journal article ↗
High Prolactin Excretion in Patients with Diabetes Mellitus and Impaired Renal Function
Triebel, J., A. I. Moreno-Vega, M. Vazquez-Membrillo, G. Nava, R. Garcia-Franco, E. Lopez-Star, O. Baldivieso-Hurtado, D. Ochoa, Y. Macotela, T. Bertsch, G. Martinez de la Escalera and C. Clapp
Clinical Laboratory 2015 · Journal article ↗ · PDF ↗
Vitamin D deficiency decreases survival of bacterial meningoencephalitis in mice
Djukic, M., N. Sostmann, T. Bertsch, M. Mecke, S. Nessler, A. Manig, U. K. Hanisch, J. Triebel, L. C. Bollheimer, C. Sieber and R. Nau
Journal of Neuroinflammation 2015 · Journal article ↗
Prolactin promotes cartilage survival and attenuates inflammation in inflammatory arthritis
Adan, N., J. Guzman-Morales, M. G. Ledesma-Colunga, S. I. Perales-Canales, A. Quintanar-Stephano, F. Lopez-Barrera, I. Mendez, B. Moreno-Carranza, J. Triebel, N. Binart, G. Martinez de la Escalera, S. Thebault and C. Clapp
Journal of Clinical Investigation 2013 · Journal article ↗ · PDF ↗
Prolactin promotes normal liver growth, survival, and regeneration in rodents: effects on hepatic IL-6, suppressor of cytokine signaling-3, and angiogenesis
Moreno-Carranza, B., M. Goya-Arce, C. Vega, N. Adan, J. Triebel, F. Lopez-Barrera, A. Quintanar-Stephano, N. Binart, G. Martinez de la Escalera and C. Clapp
American Journal of Physiology – Regulatory, Integrative and Comparative Physiology 2013 · Journal article ↗ · PDF ↗
Melanocortin receptors in rat liver cells: change of gene expression and intracellular localization during acute-phase response
Malik, I. A., J. Triebel, J. Posselt, S. Khan, P. Ramadori, D. Raddatz and G. Ramadori
Histochemistry and Cell Biology 2012 · Journal article ↗ · PDF ↗
Investigation of prolactin-related vasoinhibin in sera from patients with diabetic retinopathy
Triebel, J., M. Huefner and G. Ramadori
European Journal of Endocrinology 2009 · Journal article ↗ · PDF ↗